Properties
Description
GNE-955 is a selective and ATP-competitive Pim kinase inhibitor. It targets PIM1, PIM2, and PIM3.
Molecular Formula
C22H24N8O
Targets
PIM1: 0.018 nM (Ki); PIM2: 0.11 nM (Ki); PIM3: 0.08 nM (Ki)
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
GNE-955 can be employed in research targeting PIM kinases, focusing on its anti-tumor properties.