PKD inhibitor CID 755673, Purity ≥98%

Synonym: 521937-07-5; 7-Hydroxy-2,3,4,5-tetrahydro-1H-benzofuro[2,3-c]azepin-1-one; 2,3,4,5-Tetrahydro-7-hydroxy-1H-benzofuro[2,3-c]azepin-1-one; PKD inhibitor

MDL: MFCD03828155
CAS Number: 521937-07-5
Compound CID: 755673

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

CID 755673, soluble in DMSO and insoluble in ethanol and water, typically functions by binding to the ATP-binding site of the kinase domain, thereby preventing the phosphorylation and activation of downstream substrates. It targets PKD1, PKD2, and PKD3.

Molecular Weight

217.22

Molecular Formula

C₁₂H₁₁NO₃

Targets

PKD1: 180 nM; PKD2: 227 nM; PKD3: 280 nM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 43 mg/mL (197.95 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

CID 755673 can be used to investigate its ability to modulate specific kinase activity in biological research.