PKD inhibitor CID 755673, Purity ≥98%

Synonym: 521937-07-5; 7-Hydroxy-2,3,4,5-tetrahydro-1H-benzofuro[2,3-c]azepin-1-one; 2,3,4,5-Tetrahydro-7-hydroxy-1H-benzofuro[2,3-c]azepin-1-one; PKD inhibitor

MDL: MFCD03828155
CAS Number: 521937-07-5
Compound CID: 755673

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

CID 755673, soluble in DMSO and insoluble in ethanol and water, typically functions by binding to the ATP-binding site of the kinase domain, thereby preventing the phosphorylation and activation of downstream substrates. It targets PKD1, PKD2, and PKD3.

Molecular Weight

217.22

Molecular Formula

C₁₂H₁₁NO₃

Targets

PKD1: 180 nM; PKD2: 227 nM; PKD3: 280 nM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 43 mg/mL (197.95 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

CID 755673 can be used to investigate its ability to modulate specific kinase activity in biological research.

Storage

Store at -20ºC.