PPAR inhibitor, GSK-3787, Purity ≥98%

Synonym: 188591-46-0; GSK3787; GSK 3787; 4-Chloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide

MDL: MFCD00099612
CAS Number: 188591-46-0
Compound CID: 2800647

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

GSK-3787, soluble in DMSO and insoluble in water and ethanol, is an effective cell metabolism inhibitor, that has the ability to prevent the pathway of metabolism by inhibiting PPAR. It targets the PPARδ.

Molecular Weight

392.78

Molecular Formula

C₁₅H₁₂ClF₃N₂O₃S

Targets

PPARδ: 6.6 nM (pIC₅₀)

Form

Lyophilized powder

Purity

≥98%

Titer

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects

Solubility

In vitro: DMSO: 67 mg/mL (170.58 mM); Water: insoluble; Ethanol: insoluble

Applications

GSK-3787 is a metabolism inhibitor that can be studied extensively for its potential therapeutic applications in the treatment of various metabolic and inflammatory conditions, including diabetes and obesity.