PRMT inhibitor EPZ020411, Purity ≥98%

Synonym: 1700663-41-7; EPZ-020411; Protein arginine methyltransferase inhibitor

CAS Number: 1700663-41-7
Compound CID: 91668547

Product Size

5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

EPZ020411 inhibits enzymes that methylate arginine residues in proteins, impacting signaling pathways and gene regulation. It targets PRMT1, PRMT6, and PRMT8.

Molecular Weight

442.59

Molecular Formula

C₂₅H₃₈N₄O₃

Targets

PRMT1: 0.119 μM; PRMT6: 0.01 μM; PRMT8: 0.223 μM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

EPZ020411 can be used to inhibit the histone methyltransferase G9a, aiding epigenetic research.

Storage

Store at -20ºC.