Properties
Description
MS049 inhibits enzymes that methylate arginine residues in proteins, impacting signaling pathways and gene regulation. It targets PRMT4, PRMT6, and PRMT8.
Molecular Formula
C15H24N2O
Targets
PRMT4: 34 nM; PRMT6: 43 nM (); PRMT8: 1600 nM
Identity
Confirmed by NMR/HPLC/MS.
Applications
MS049 can be applied in research focused on the selective inhibition of protein arginine methyltransferase 4 (PRMT4/CARM1).