R-268712

Synonym: 879487-87-3; 2-[4-[2-Fluoro-5-[3-(6-methylpyridine-2-yl)-1H-pyrazol-4-yl] phenyl] pyrazol-1-yl]ethanol

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

R-268712 inhibits the activity of protein-tyrosine kinases that play a critical role in cell signaling and regulation. It targets Smad3, and TGFBR1.

Molecular Weight

363.39

Molecular Formula

C₂₀H₁₈FN₅O

Targets

Smad3: 10.4 nM; TGFBR1: 2.5 nM

Form

Lyophilized powder

Purity

>98%

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

R-268712 can be used for its ability to inhibit these abnormally activated enzymes that disrupt pathological processes.

Storage

Store at -20℃, and keep desiccated.