Properties
Description
Roluperidone inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT2A receptor, and Sigma-2 receptor.
Molecular Formula
C22H23FN2O2
Targets
5-HT2A receptor: 7.53 nM; Sigma-2 receptor: 8.19 nM
Applications
Roluperidone can be used for research on hallucinations, delusions, disorganized thinking, and negative symptoms.