Properties
Description
RS-127445, soluble in DMSO and ethanol and insoluble in water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT2B, and 5-HT2B.
Molecular Formula
C17H16FN3
Targets
5-HT2B: 10.4(pIC50); 5-HT2B: 9.5 (pKi)
Solubility
DMSO: 54 mg/mL (191.94 mM); Water: insoluble; Ethanol: 8 mg/mL (28.43 mM)
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
RS-127445 can be used to research various conditions related to the serotonin system and its receptors.
Storage
Store at -20°C, and keep desiccated.