Properties
Description
Rupatadine Fumarate inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets histamine H1 receptor, and PAFR.
Molecular Formula
C26H26ClN3·C4H4O4
Targets
Histamine H1 receptor: 102 nM (Ki); PAFR: 550 nM (Ki)
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
Rupatadine fumarate can be studied for its effect on blocking the activity of dopamine receptors in the brain, which are believed to play a role in the development of psychotic symptoms.
Storage
Store at -20°C, and keep desiccated.
