Properties
Description
S1RA (E-52862), soluble in DMSO, ethanol and water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets sigma 1 receptor.
Molecular Formula
C20H23N3O2
Targets
Sigma 1 receptor: 17nM
Solubility
DMSO: 63 mg/mL (186.71 mM); Water: 63 mg/mL (186.71 mM); Ethanol: 18 mg/mL (53.34 mM)
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
S1RA can be used for its antidepressant and anxiolytic effects.
Storage
Store at -20°C, and keep desiccated.
