Properties
Description
Sarpogrelate hydrochloride, soluble in DMSO, ethanol and water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT2A receptor, 5-HT2B receptor, and 5-HT2C receptor.
Molecular Formula
C24H32ClNO6
Targets
5-HT2A receptor: 8.52 (pKi); 5-HT2B receptor: 6.57 (pKi); 5-HT2C receptor: 7.43 (pKi)
Solubility
DMSO: 92 mg/mL (197.43 mM); Water: 92 mg/mL (197.43 mM); Ethanol: 30 mg/mL (64.38 mM)
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
Sarpogrelate hydrochloride can be studied for its effect on inhibiting the action of serotonin on blood vessels.
Storage
Store at -20°C, and keep desiccated.
