Seltorexant

Synonym: 1293281-49-8; 2-{5-[2-Fluoro-6-(2H-1,2,3-triazol-2-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrol-2-yl}-4,6-dimethylpyrimidine

Product Size

1 mg; 5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Seltorexant inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets human OX2R, and rat OX2R.

Molecular Weight

407.44

Molecular Formula

C₂₁H₂₂FN₇O

Targets

Human OX2R: 8.0 (pKi); Rat OX2R: 8.1 (pKi)

Form

Lyophilized powder

Purity

>98%

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

Seltorexant can be studied for its effect on blocking the action of orexin, a neuropeptide involved in the regulation of wakefulness and sleep.

Storage

Store at -20°C, and keep desiccated.