Properties
Description
RQ-00203078 modulates the function of TRP channels, which are crucial for various physiological processes including sensation and thermoregulation. It targets TRPM8, TRPM8, and TRPV4.
Molecular Formula
C21H13ClF6N2O5S
Targets
TRPM8: 5.3 nM; TRPM8: 8.3 nM (IC50, human TRPM8 channels); TRPV4: 10 μM
Identity
Confirmed by NMR/HPLC/MS.
Applications
RQ-00203078 is investigated as a TRP channel inhibitor, aiming to understand its role in sensory and pain processing pathways.
