TRPV inhibitor AMG517, Purity ≥98%

Synonym: 659730-32-2; TRPV inhibitor; AMG 517; AMG-517

MDL: MFCD14584859
CAS Number: 659730-32-2
Compound CID: 16007367

Product Size

5 mg; 10 mg; 25 mg; 50 mg

Price

Datasheet

MSDS

Properties

Description

AMG517, soluble in DMSO and insoluble in ethanol and water, blocks the activity of transient receptor potential vanilloid channels, often used to study pain mechanisms. It targets TRPV1.

Molecular Weight

430.4

Molecular Formula

C₂₀H₁₃F₃N₄O₂S

Targets

TRPV1: 1-2 nM

Form

Lyophilized powder

Purity

Solubility

DMSO: 84 mg/mL (195.16 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

AMG517 is a TRPV1 channel inhibitor used in the study of pain and inflammatory responses.