TRPV inhibitor SB-705498, Purity ≥98%

Synonym: 501951-42-4; TRPV inhibitor; SB705498

MDL: MFCD13152399
CAS Number: 501951-42-4
Compound CID: 9910486

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

SB-705498, soluble in DMSO and ethanol and insoluble in water, blocks the activity of transient receptor potential vanilloid channels, often used to study pain mechanisms. It targets hTRPV1 and hTRPV1.

Molecular Weight

428

Molecular Formula

C₁₇H₁₆BrF₃N₄O

Targets

hTRPV1: 7.6 (pKi); hTRPV1: 7.1(pIC₅₀)

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 78 mg/mL (181.71 mM); Water: Insoluble; Ethanol: 18 mg/mL (41.93 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

SB-705498 is a TRPV (transient receptor potential vanilloid) channel inhibitor used in research to explore pain pathways and treatment through modulation of these channels.