Urapidil hydrochloride

Synonym: 64887-14-5; Urapidil HCl

CAS Number: 64887-14-5
Compound CID: 167980

Product Size

100 mg; 200 mg; 500 mg; 1 g

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Urapidil hydrochloride, soluble in DMSO, ethanol and water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets α adrenergic receptor, α1-adrenergic receptor, α2-adrenergic receptor, and 5-HT1A receptor.

Molecular Weight

423.94

Molecular Formula

C₂₀H₂₉N₅O₃·HCl

Targets

α Adrenergic receptor; α1-Adrenergic receptor: 6.13 (pIC₅₀); α2-Adrenergic receptor: 4.38 (pIC₅₀); 5-HT1A receptor

Form

Lyophilized powder

Purity

>98%

Solubility

DMSO: 23 mg/mL (54.25 mM); Water: 81 mg/mL (191.06 mM); Ethanol: 1 mg/mL (2.35 mM)

Applications

Urapidil hydrochloride can be used to research and develop therapeutic strategies for certain diseases that involve excessive activation of GPCR-G protein signaling pathways.