Properties
Description
TG 100801 HCl is a protein tyrosine kinase inhibitor that has shown potent biochemical activity against VEGFR. It targets FGFR1, FGFR2, PDGFRβ, VEGFR1, and VEGFR2.
Molecular Formula
C33H31Cl2N5O3
Targets
FGFR1: 2 nM; FGFR2: 16 nM; PDGFRβ: 13 nM; VEGFR1: 2 nM; VEGFR2: 7 nM
Identity
Confirmed by NMR/HPLC/MS.
Applications
TG 100801 HCl is used in research focusing on blocking VEGFR, which is vital for anti-cancer therapy studies.