Casein kinase inhibitor TBB, Purity ≥98%

Synonym: 17374-26-4; Casein kinase inhibitor; NSC 231634

MDL: MFCD06411399
CAS Number: 17374-26-4
Compound CID: 1694

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

TBB, soluble in DMSO, is a potent compound that inhibits Casein kinase activity. It targets CDK2, CK2, DYRK1a, DYRK2, DYRK3, HIPK2, HIPK3, PIM1, PIM2, PIM3, and PKD1.

Molecular Weight

434.71

Molecular Formula

C₆HBr₄N₃

Targets

CDK2: 14 μM; CK2: 0.15 μM (human CK2); DYRK1a: 4.36 μM; DYRK2: 0.99 μM; DYRK3: 5.3 μM; HIPK2: 5.3 μM; HIPK3: 4.9 μM; PIM1: 1.04 μM; PIM2: 4.3 μM; PIM3: 0.86 μM; PKD1: 5.9 μM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 78 mg/mL (179.43 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

TBB is a Casein kinase inhibitor used in research to explore its potential in regulating cellular processes such as inflammation and cancer.